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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TQ0084 | Lumateperone Tosylate | ITI-007 | Dopamine Receptor , 5-HT Receptor |
lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist (Ki: 0.54 nM), a SERT blocker (Ki: 61 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki: 32 nM). | |||
T21069 | Lumateperone | ITI 722,ITI722,ITI-007,ITI007 | 5-HT Receptor |
Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM). | |||
T2226 | Pergolide mesylate | Pergolide mesylate salt,LY127809,Pergolide methanesulfonate | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor |
Pergolide mesylate salt(LY127809) is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due to potential for HEART VALVE DISEASES. | |||
T0302 | Triflupromazine hydrochloride | Neoprin,Fluopromazine hydrochloride,Fluorofen,Flumazin | Dopamine Receptor , 5-HT Receptor , AChR , Autophagy |
Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists. | |||
T6988 | SKF 38393 hydrochloride | (±)-SKF-38393 hydrochloride,SKF-38393A,SKF38393 HCl | Dopamine Receptor |
SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1/D5 receptor agonist. | |||
T16999 | Tavapadon | PF-6649751,CVL-751 | Dopamine Receptor |
Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist. | |||
T21782 | A 77636 hydrochloride | A77636 hydrochloride | Dopamine Receptor |
A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM). A 77636 hydrochloride shows antiparkinsonian activity. A 77636 hydrochloride is functionall... | |||
T6648 | Rotundine | Gindarine,L-Tetrahydropalmatine,Caseanine,(-)-Tetrahydropalmatine | Dopamine Receptor , 5-HT Receptor |
Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM. | |||
T67729 | UCM-1306 | Dopamine Receptor | |
UCM-1306 is a potent and orally active allosteric modulator (PAM) of human dopamine D1 receptor. UCM-1306 could increase the maximal effect of endogenous dopamine (DA) both in human and mouse D1 receptors. UCM-1306 could... | |||
T8702 | SKF-83566 | Dopamine Receptor , 5-HT Receptor , AChR | |
SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 nM | |||
T2564 | Cis-(Z)-Flupentixol dihydrochloride | Emergil,Flupenthixol dihydrochloride | Dopamine Receptor , 5-HT Receptor |
cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist. | |||
T22921 | LE 300 | Dopamine Receptor , 5-HT Receptor | |
dopamine D1 receptor antagonist | |||
T4369 | SCH-23390 hydrochloride | R-(+)-SCH23390 hydrochloride | Potassium Channel , Dopamine Receptor , 5-HT Receptor |
SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM). | |||
T14767 | BP 897 hydrochloride | Dopamine Receptor | |
BP 897 is a potent and selective agonist of dopamine D3 receptor and it is a weak dopamine D2 receptor antagonist, with Kis of 0.92 nM and 61 nM for D3 and D2 receptors. Which shows low affinities at D1 and D4 receptors ... | |||
T60835 | SKF83959 | Dopamine Receptor | |
SKF83959, a benzazepine analog, is a selective and potent partial agonist of the dopamine D1 receptor with Ki values of 1.18, 7.56, 920, and 399 nM for rat D1, D5, D2, and D3 receptors, respectively.SKF83959 is a potent ... | |||
T4274 | Melitracen hydrochloride | Thymeol hydrochloride,Melixeran | Dopamine Receptor , 5-HT Receptor |
Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression. | |||
T6835 | Fenoldopam mesylate | Fenoldopam methanesulfonate,SKF-82526 mesylate,Corlopam mesylate,mesylate,SKF 82526 | Dopamine Receptor |
Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties. It lowers blood pressure through arteriolar vasodilation. | |||
T9100 | BP 897 | 2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]- | Dopamine Receptor |
BP 897 (2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-) is a potent and selective dopamine D3 receptor agonist, and a weak dopamine D2 receptor antagonist, with Kis of 0.92 nM and 61 nM for D3 ... | |||
T21446 | Rotigotine Hydrochloride | Rotigotine (Hydrochloride),N 0923,N-0924,Rotigotine HCl,N-0923 | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor |
Rotigotine Hydrochloride (N-0924), a dopamine receptor agonist prefering for D3 receptors over D1 and D2, has effective activity of anti-Parkinsonian. Racemic rotigotine hydrochloride is about 50 times as potent as quinp... | |||
T28167 | NGB 2904 | NGB2904 HCl,NGB-2904,NGB2904 | Others , Dopamine Receptor , 5-HT Receptor |
NGB 2904 is a potent and selective antagonist of dopamine D3 receptor (Ki values are 1.4, 217, 223, 642, > 5000, > 10000 and > 10000 nM for D3, D2, 5-HT2, α1, D4, D1 and D5 receptors respectively). NGB2904 potently antag... |